TargetMol

C-82

Product Code:
 
TAR-T10641
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10641-1mg1mg£434.00
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TAR-T10641-5mg5mg£804.00
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Quantity:
TAR-T10641-1mL1 mL * 10 mM (in DMSO)£1,026.00
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TAR-T10641-10mg10mg£1,130.00
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Quantity:
TAR-T10641-25mg25mg£1,749.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
C-82 is a specific CBP/β-catenin antagonist. It inhibits the binding between β-catenin and CBP and increases the binding between β-catenin and p300.
CAS:
1422253-37-9
Formula:
C33H34N6O4
Molecular Weight:
578.673
Pathway:
Chromatin/Epigenetic; Stem Cells; Cytoskeletal Signaling
Purity:
0.9966
SMILES:
[H][C@]12[C@H](C)N(Cc3cccc4cccnc34)C(=O)[C@H](Cc3ccc(O)cc3)N1C(=O)CN(C)N2C(=O)NCc1ccccc1
Target:
Epigenetic Reader Domain; Wnt/beta-catenin

References

1. Osawa Y, et al. Inhibition of Cyclic Adenosine Monophosphate (cAMP)-response Element-binding Protein (CREB)-binding Protein (CBP)/?-Catenin Reduces Liver Fibrosis in Mice. EBioMedicine. 2015 Oct 8;2(11):1751-8.