TargetMol

DDP-38003 trihydrochloride

Product Code:
 
TAR-T10983
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10983-100mg100mg£1,332.00
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Further Information

Bioactivity:
DDP-38003 trihydrochloride is a novel, orally available histone lysine specific demethylase 1A (KDM1A / LSD1) inhibitor with IC50 of 84 nM.
CAS:
T10983
Formula:
C21H29Cl3N4O
Molecular Weight:
459.84
Purity:
0.98
SMILES:
[H]Cl.[H]Cl.O=C(NC1=CC=C([C@@H]2C[C@H]2N)C=C1)C(C=C3)=CC=C3N4CCN(C)CC4.[H]Cl

References

1. Vianello P, et al. Discovery of a Novel Inhibitor of Histone Lysine-Specific Demethylase 1A (KDM1A/LSD1) as Orally Active Antitumor Agent. J Med Chem. 2016 Feb 25;59(4):1501-17.