TargetMol

Elenbecestat

Product Code:
 
TAR-T11175
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11175-1mg1mg£122.00
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TAR-T11175-5mg5mg£195.00
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TAR-T11175-1mL1 mL * 10 mM (in DMSO)£206.00
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TAR-T11175-10mg10mg£282.00
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TAR-T11175-25mg25mg£510.00
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TAR-T11175-50mg50mg£704.00
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Quantity:
TAR-T11175-100mg100mg£938.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Elenbecestat is an effective oral bioutilization and CNS penetrating ACE-1 inhibitor for the treatment of Alzheimer's disease.
CAS:
1388651-30-6
Formula:
C19H18F3N5O2S
Molecular Weight:
437.44
Pathway:
Neuroscience
Purity:
0.9967
SMILES:
[H][C@]12CSC(N)=N[C@]1(CO[C@@H]2C)c1cc(NC(=O)c2cnc(cn2)C(F)F)ccc1F
Target:
Beta-Secretase; BACE

References

1. Kumar D, et al.Secretase inhibitors for the treatment of Alzheimer's disease: Long road ahead. Eur J Med Chem. 2018 Mar 25;148:436-452. 2. A single dose of the beta-secretase inhibitor, e2609, decreases CSF bace1 enzymatic activity in cynomolgus monkeys. Alzheimer?s & Dementia, 8(4), P224.