TargetMol

EPAC 5376753

Product Code:
 
TAR-T11212
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11212-1mg1mg£148.00
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TAR-T11212-5mg5mg£245.00
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TAR-T11212-10mg10mg£324.00
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TAR-T11212-25mg25mg£498.00
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Quantity:
TAR-T11212-50mg50mg£688.00
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This product comes from: United States.
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Further Information

Bioactivity:
EPAC 5376753 is an allosteric inhibitor of EPAC1 with an IC50 of 4 ?M in Swiss 3T3 cells.
CAS:
302826-61-5
Formula:
C15H8Cl2N2O3S
Molecular Weight:
367.2
Pathway:
GPCR/G Protein
Purity:
0.98
SMILES:
Clc1ccc(-c2ccc(C=C3C(=O)NC(=S)NC3=O)o2)c(Cl)c1
Target:
cAMP

References

1. Brown LM, et al. Allosteric inhibition of Epac: computational modeling and experimental validation to identify allosteric sites and inhibitors. J Biol Chem. 2014 Oct 17;289(42):29148-57.