TargetMol

ERAP1-IN-1

Product Code:
 
TAR-T11221
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11221-1mg1mg£179.00
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Quantity:
TAR-T11221-1mL1 mL * 10 mM (in DMSO)£303.00
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Quantity:
TAR-T11221-5mg5mg£303.00
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Quantity:
TAR-T11221-10mg10mg£454.00
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Quantity:
TAR-T11221-25mg25mg£704.00
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Quantity:
TAR-T11221-50mg50mg£938.00
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Quantity:
TAR-T11221-100mg100mg£1,259.00
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Quantity:
TAR-T11221-500mg500mg£2,456.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 allosterically activates ERAP1?s hydrolysis of fluorogenic and chromogenic amino acid substrates but competitively inhibits its activity toward a nonamer peptide representative of physiological substrates.
CAS:
865273-97-8
Formula:
C20H21F3N2O5S
Molecular Weight:
458.45
Purity:
0.986
SMILES:
COc1ccc(cc1S(=O)(=O)Nc1cc(ccc1N1CCCCC1)C(F)(F)F)C(O)=O

References

1. Maben Z, et al. Discovery of Selective Inhibitors of Endoplasmic Reticulum Aminopeptidase 1. J Med Chem. 2019 Dec 30.