TargetMol

GPI-1046

Product Code:
 
TAR-T11451
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T11451-1mg1mg£125.00
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TAR-T11451-2mg2mg£147.00
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TAR-T11451-1mL1 mL * 10 mM (in DMSO)£177.00
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TAR-T11451-5mg5mg£189.00
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TAR-T11451-10mg10mg£269.00
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TAR-T11451-25mg25mg£406.00
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TAR-T11451-50mg50mg£549.00
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TAR-T11451-100mg100mg£764.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GPI-1046 is an immunophilin ligand without antibiotic action and attenuates ethanol intake in part through the upregulation of glutamate transporter 1 (GLT1) in PFC and NAc-core.
CAS:
186452-09-5
Formula:
C20H28N2O4
Molecular Weight:
360.45
Pathway:
Proteases/Proteasome; ; Microbiology/Virology
Purity:
0.9991
SMILES:
O=C(OCCCC1=CC=CN=C1)[C@H]2N(C(C(C(C)(C)CC)=O)=O)CCC2
Target:
HIV Protease

References

1. Sari Y, et al. Neuroimmunophilin GPI-1046 reduces ethanol consumption in part through activation of GLT1 in alcohol-preferring rats. Neuroscience. 2012 Dec 27;227:327-35. 2. Eberling JL, et al. The immunophilin ligand GPI-1046 does not have neuroregenerative effects in MPTP-treated monkeys. Exp Neurol. 2002 Dec;178(2):236-42.