TargetMol

HA155

Product Code:
 
TAR-T11533
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11533-1mg1mg£168.00
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TAR-T11533-5mg5mg£369.00
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TAR-T11533-1mL1 mL * 10 mM (in DMSO)£375.00
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TAR-T11533-10mg10mg£511.00
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TAR-T11533-25mg25mg£768.00
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TAR-T11533-50mg50mg£1,010.00
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Quantity:
TAR-T11533-100mg100mg£1,340.00
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This product comes from: United States.
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Further Information

Bioactivity:
HA155 selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.
CAS:
1312201-00-5
Formula:
C24H19BFNO5S
Molecular Weight:
463.29
Pathway:
Metabolism
Purity:
0.9828
SMILES:
O=C1N(CC2=CC=C(F)C=C2)C(S/C1=CC3=CC=C(OCC4=CC=C(B(O)O)C=C4)C=C3)=O.[(Z)]
Target:
PDE

References

1. Albers HM, et al. Structure-based design of novel boronic acid-based inhibitors of autotaxin. J Med Chem. 2011 Jul 14;54(13):4619-26. 2. Fulkerson Z, et al. Binding of autotaxin to integrins localizes lysophosphatidic acid production to platelets and mammalian cells. J Biol Chem. 2011 Oct 7;286(40):34654-63. 3. Albers HM, et al. Chemical Evolution of Autotaxin Inhibitors. Chem Rev. 2012 May 9;112(5):2593-603.