TargetMol

OMDM-5

Product Code:
 
TAR-T12306
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12306-1mg1mg£189.00
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TAR-T12306-5mg5mg£340.00
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TAR-T12306-1mL1 mL * 10 mM (in DMSO)£382.00
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TAR-T12306-10mg10mg£470.00
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TAR-T12306-25mg25mg£707.00
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TAR-T12306-50mg50mg£978.00
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TAR-T12306-100mg100mg£1,291.00
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TAR-T12306-500mg500mg£2,456.00
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Further Information

Bioactivity:
OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing weak ligand activity at cannabinoid type 1 receptor (CB1, Ki=4.9 μM). OMDM-5 is a selective anandamide cellular uptake (ACU) inhibitor(Ki = 4.8 μM).
CAS:
616884-66-3
Formula:
C26H44N2O3
Molecular Weight:
432.649
Pathway:
GPCR/G Protein; Membrane transporter/Ion channel; Metabolism
Purity:
0.9972
SMILES:
CCCCCCCCC=C/CCCCCCCC(=O)NNCc1ccc(O)c(OC)c1
Target:
Cannabinoid Receptor; Endogenous Metabolite; TRP/TRPV Channel

References

1. Ortar G, et al. Novel selective and metabolically stable inhibitors of anandamide cellular uptake. Biochem Pharmacol. 2003 May 1;65(9):1473-81.