TargetMol

Sigma-1 receptor antagonist 1

Product Code:
 
TAR-T12910
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12910-1mg1mg£148.00
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TAR-T12910-5mg5mg£269.00
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TAR-T12910-1mL1 mL * 10 mM (in DMSO)£320.00
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TAR-T12910-10mg10mg£389.00
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TAR-T12910-25mg25mg£603.00
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TAR-T12910-50mg50mg£830.00
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TAR-T12910-100mg100mg£1,099.00
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TAR-T12910-500mg500mg£2,135.00
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Further Information

Bioactivity:
Sigma-1 receptor antagonist 1 is an effective and selective antagonist of sigma-1 receptor. Sigma-1 receptor antagonist 1 exhibits antineuropathic pain activity and can be used in the treatment of neuropathic pain studies.
CAS:
1639220-19-1
Formula:
C19H23Cl2N3O
Molecular Weight:
380.31
Pathway:
GPCR/G Protein
Purity:
0.9981
SMILES:
Cc1nc(nc(OCCCN2CCCCC2)c1Cl)-c1ccc(Cl)cc1
Target:
Sigma receptor

References

1. Lan Y, et al. Synthesis and biological evaluation of novel sigma-1 receptor antagonists based on pyrimidine scaffold as agents for treating neuropathic pain. J Med Chem. 2014 Dec 26;57(24):10404-23.