TargetMol

Src Inhibitor 3

Product Code:
 
TAR-T13000
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13000-1mg1mg£195.00
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TAR-T13000-5mg5mg£334.00
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TAR-T13000-1mL1 mL * 10 mM (in DMSO)£463.00
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TAR-T13000-10mg10mg£523.00
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TAR-T13000-25mg25mg£785.00
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TAR-T13000-50mg50mg£1,058.00
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Quantity:
TAR-T13000-100mg100mg£1,412.00
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Further Information

Bioactivity:
Src Inhibitor 3 is an effective inhibitor of c-terminal Src kinase (IC50 <3 nM in CSK HTRF, <4 nM in Caliper assay). Src Inhibitor 3 increases T cell proliferation induced by T cell receptor signaling.
CAS:
2380027-49-4
Formula:
C34H32ClFN8O4
Molecular Weight:
671.13
Pathway:
; Angiogenesis; Tyrosine Kinase/Adaptors
Purity:
0.98
SMILES:
COc1ccc2c(cnn2c1)C(=O)Nc1ccc(NC(=O)c2nn(C3CCN(CC3)C(=O)CC(C)(C)C#N)c3ccc(F)cc23)cc1Cl
Target:
Src

References

1. O'Malley DP, et al. Discovery of Pyridazinone and Pyrazolo[1,5-a]pyridine Inhibitors of C-Terminal Src Kinase. ACS Med Chem Lett. 2019 Sep 25;10(10):1486-1491.