TargetMol

EHP-101

Product Code:
 
TAR-T13289
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T13289-1mg1mg£158.00
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Quantity:
TAR-T13289-5mg5mg£262.00
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Quantity:
TAR-T13289-1mL1 mL * 10 mM (in DMSO)£282.00
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TAR-T13289-10mg10mg£389.00
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Quantity:
TAR-T13289-25mg25mg£594.00
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Quantity:
TAR-T13289-50mg50mg£804.00
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Quantity:
TAR-T13289-100mg100mg£1,058.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
VCE-004.8 is a specific dual agonist of PPARγ and CB2 receptor with potent anti-inflammatory activity. VCE-004.8 attenuates adipogenesis and prevents diet-induced obesity.
CAS:
1818428-24-8
Formula:
C28H35NO3
Molecular Weight:
433.592
Pathway:
Metabolism; GPCR/G Protein; Chromatin/Epigenetic; DNA Damage/DNA Repair
Purity:
0.98
SMILES:
CCCCCC1=C(NCc2ccccc2)C(=O)C([C@@H]2C=C(C)CC[C@H]2C(C)=C)=C(O)C1=O
Target:
Cannabinoid Receptor; HIF/HIF Prolyl-Hydroxylase; PPAR

References

1. Navarrete C, et al. Hypoxia mimetic activity of VCE-004.8, a cannabidiol quinone derivative: implications for multiple sclerosis therapy. J Neuroinflammation. 2018 Mar 1;15(1):64. 2. Palomares B, et al. VCE-004.8, A Multitarget Cannabinoquinone, Attenuates Adipogenesis and Prevents Diet-Induced Obesity. Sci Rep. 2018 Oct 31;8(1):16092.