TargetMol

WS-383

Product Code:
 
TAR-T13349
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13349-1mg1mg£101.00
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TAR-T13349-2mg2mg£113.00
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TAR-T13349-5mg5mg£142.00
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TAR-T13349-1mL1 mL * 10 mM (in DMSO)£149.00
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TAR-T13349-10mg10mg£189.00
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TAR-T13349-25mg25mg£309.00
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TAR-T13349-50mg50mg£543.00
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TAR-T13349-100mg100mg£744.00
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TAR-T13349-500mg500mg£1,452.00
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Further Information

Bioactivity:
WS-383 is a selective, potent and reversible DCN1-UBC12 interaction inhibitor(IC50 of 11 nM).
CAS:
2247544-02-9
Formula:
C18H21Cl2N9S2
Molecular Weight:
498.45
Pathway:
Ubiquitination
Purity:
0.988
SMILES:
Cl.CN(C)CCn1nnnc1Sc1cc(C)nc2nc(SCc3ccc(Cl)cc3)nn12
Target:
E1/E2/E3 Enzyme

References

1. Wang S, et al. Development of Highly Potent, Selective, and Cellular Active Triazolo[1,5- a]pyrimidine-Based Inhibitors Targeting the DCN1-UBC12 Protein-Protein Interaction. J Med Chem. 2019 Mar 14;62(5):2772-2797.