TargetMol

Elacestrant

Product Code:
 
TAR-T13674
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13674-1mg1mg£189.00
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TAR-T13674-5mg5mg£349.00
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TAR-T13674-1mL1 mL * 10 mM (in DMSO)£382.00
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TAR-T13674-10mg10mg£470.00
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TAR-T13674-25mg25mg£707.00
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TAR-T13674-50mg50mg£978.00
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TAR-T13674-100mg100mg£1,291.00
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This product comes from: United States.
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Further Information

Bioactivity:
Elacestrant with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant ?is an orally available selective estrogen receptor degrader .
CAS:
722533-56-4
Formula:
C30H38N2O2
Molecular Weight:
458.646
Pathway:
Endocrinology/Hormones
Purity:
0.9892
SMILES:
CCNCCc1ccc(CN(CC)c2cc(OC)ccc2[C@@H]2CCc3cc(O)ccc3C2)cc1
Target:
Estrogen Receptor/ERR; Estrogen/progestogen Receptor

References

1. Garner F, et al. RAD1901: a novel, orally bioavailable selective estrogen receptor degrader that demonstrates antitumor activity in breast cancer xenograft models. Anticancer Drugs. 2015 Oct;26(9):948-56.