TargetMol

GSK1379725A

Product Code:
 
TAR-T15424
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T15424-1mg1mg£160.00
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TAR-T15424-5mg5mg£229.00
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TAR-T15424-1mL1 mL * 10 mM (in DMSO)£252.00
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TAR-T15424-10mg10mg£349.00
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TAR-T15424-25mg25mg£544.00
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TAR-T15424-50mg50mg£747.00
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Quantity:
TAR-T15424-100mg100mg£1,002.00
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Quantity:
TAR-T15424-500mg500mg£1,942.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GSK1379725A is a selective BPTF ligand (Kd = 2.8 μM).
CAS:
1802251-00-8
Formula:
C23H23FN6O3
Molecular Weight:
450.474
Pathway:
Chromatin/Epigenetic
Purity:
0.9959
SMILES:
COC(=O)c1cccc(NC(=O)NC2CCN(C2)c2ccnc(Nc3ccc(F)cc3)n2)c1
Target:
Epigenetic Reader Domain

References

1. Urick AK, et al. Dual Screening of BPTF and Brd4 Using Protein-Observed Fluorine NMR Uncovers New Bromodomain Probe Molecules. ACS Chem Biol. 2015 Oct 16;10(10):2246-56.