TargetMol

LY2955303

Product Code:
 
TAR-T15811
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15811-50mg50mg£466.00
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Further Information

Bioactivity:
LY2955303 is an effective and selective antagonist of retinoic acid receptor gamma (RARγ, Ki = 1.09 nM).
CAS:
1433497-19-8
Formula:
C36H42N4O3
Molecular Weight:
578.757
Pathway:
Metabolism;
Purity:
0.9856
SMILES:
CN1CCN(CC1)C(=O)c1ccc(cc1)-n1nc(cc1-c1cc(cc(c1)C(C)(C)C)C(C)(C)C)-c1ccc(cc1)C(O)=O
Target:
Retinoid Receptor

References

1. Hughes NE, et al. Identification of potent and selective retinoic acid receptor gamma (RAR?) antagonists for the treatment of osteoarthritis pain using structure based drug design. Bioorg Med Chem Lett. 2016 Jul 15;26(14):3274-3277.