TargetMol

Islatravir

Product Code:
 
TAR-T16098
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16098-1mg1mg£201.00
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TAR-T16098-5mg5mg£349.00
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TAR-T16098-1mL1 mL * 10 mM (in DMSO)£499.00
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TAR-T16098-10mg10mg£523.00
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TAR-T16098-25mg25mg£785.00
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TAR-T16098-50mg50mg£1,058.00
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Quantity:
TAR-T16098-100mg100mg£1,412.00
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This product comes from: United States.
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Further Information

Bioactivity:
Islatravir is an effective anti-HIV-1 agent. It acts as a nucleoside reverse transcriptase inhibitor (EC50s: 0.068 nM, 3.1 nM, and 0.15 nM for HIV-1 (WT), HIV-1 (M184V), HIV-1 (MDR), respectively).
CAS:
865363-93-5
Formula:
C12H12FN5O3
Molecular Weight:
293.258
Pathway:
Microbiology/Virology; Proteases/Proteasome
Purity:
0.9703
SMILES:
Nc1nc(F)nc2n(cnc12)[C@H]1C[C@H](O)[C@@](CO)(O1)C#C
Target:
HIV Protease; Reverse Transcriptase

References

1. Ohrui H, et al. 2'-deoxy-4'-C-ethynyl-2-fluoroadenosine, a nucleoside reverse transcriptase inhibitor, is highly potent against all human immunodeficiency viruses type 1 and has low toxicity. Chem Rec. 2006;6(3):133-43.