TargetMol

MPI_5a

Product Code:
 
TAR-T16129
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16129-1mg1mg£294.00
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TAR-T16129-2mg2mg£428.00
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TAR-T16129-1mL1 mL * 10 mM (in DMSO)£650.00
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TAR-T16129-5mg5mg£744.00
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TAR-T16129-10mg10mg£978.00
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TAR-T16129-25mg25mg£1,412.00
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Quantity:
TAR-T16129-50mg50mg£1,886.00
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TAR-T16129-100mg100mg£2,456.00
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Further Information

Bioactivity:
MPI_5a is an effective and selective inhibitor of HDAC6 (IC50=36 nM). MPI_5a weakly inhibits other HDAC isoforms and it also inhibits acyl-tubulin accumulation in cells (IC50: 210 nM).
CAS:
1259296-46-2
Formula:
C16H17N3O3
Molecular Weight:
299.33
Pathway:
Chromatin/Epigenetic; DNA Damage/DNA Repair
Purity:
0.98
SMILES:
Cn1cccc1C(=O)N1CCc2cc(ccc2C1)C(=O)NO
Target:
HDAC

References

1. Blackburn C, et al. Potent histone deacetylase inhibitors derived from 4-(aminomethyl)-N-hydroxybenzamide with high selectivity for the HDAC6 isoform. J Med Chem. 2013 Sep 26;56(18):7201-11.