TargetMol

SBI-553

Product Code:
 
TAR-T16860
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16860-1mg1mg£179.00
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TAR-T16860-5mg5mg£303.00
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TAR-T16860-1mL1 mL * 10 mM (in DMSO)£326.00
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TAR-T16860-10mg10mg£436.00
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TAR-T16860-25mg25mg£675.00
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TAR-T16860-50mg50mg£922.00
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Quantity:
TAR-T16860-100mg100mg£1,219.00
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This product comes from: United States.
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Further Information

Bioactivity:
SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).
CAS:
1849603-72-0
Formula:
C26H31FN4O2
Molecular Weight:
450.558
Pathway:
GPCR/G Protein
Purity:
0.9969
SMILES:
COc1ccccc1C1CCN(CC1)c1nc(nc2ccc(cc12)N(C)CCO)C1(F)CC1
Target:
Neurotensin Receptor

References

1. Pinkerton AB, et al. Discovery of ?-Arrestin Biased, Orally Bioavailable, and CNS Penetrant Neurotensin Receptor 1 (NTR1) Allosteric Modulators. J Med Chem. 2019 Aug 20.