TargetMol

Tegoprazan

Product Code:
 
TAR-T17030
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T17030-1mg1mg£123.00
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TAR-T17030-5mg5mg£198.00
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TAR-T17030-1mL1 mL * 10 mM (in DMSO)£212.00
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TAR-T17030-10mg10mg£275.00
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TAR-T17030-25mg25mg£483.00
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TAR-T17030-50mg50mg£724.00
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TAR-T17030-100mg100mg£1,058.00
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TAR-T17030-200mg200mg£1,420.00
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Further Information

Bioactivity:
Tegoprazan is a potassium-competitive acid blocker and is a potent, oral active, and highly selective inhibitor of gastric H+/K+-ATPase. That could control gastric acid secretion and motility (IC50: ranging from 0.29-0.52 μM for porcine, canine, and human H+/K+-ATPases in vitro).
CAS:
942195-55-3
Formula:
C20H19F2N3O3
Molecular Weight:
387.387
Pathway:
Membrane transporter/Ion channel
Purity:
0.9822
SMILES:
CN(C)C(=O)c1cc(O[C@H]2CCOc3cc(F)cc(F)c23)c2nc(C)[nH]c2c1
Target:
ATPase; Proton pump

References

1. Takahashi N, et al. Tegoprazan, a Novel Potassium-Competitive Acid Blocker to Control Gastric Acid Secretion and Motility. J Pharmacol Exp Ther. 2018 Feb;364(2):275-286.