TargetMol

Endoxifen (Z-isomer)

Product Code:
 
TAR-T2280
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T2280-1mg1mg£115.00
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TAR-T2280-2mg2mg£136.00
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TAR-T2280-1mL1 mL * 10 mM (in DMSO)£169.00
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TAR-T2280-5mg5mg£177.00
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TAR-T2280-10mg10mg£242.00
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TAR-T2280-25mg25mg£389.00
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Quantity:
TAR-T2280-50mg50mg£566.00
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This product comes from: United States.
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Further Information

Bioactivity:
Endoxifen (EDX) is a key active metabolite of tamoxifen (TAM) with higher affinity and specificity to estrogen receptors that also inhibits aromatase activity.
CAS:
112093-28-4
Formula:
C25H27NO2
Molecular Weight:
373.496
Pathway:
Tyrosine Kinase/Adaptors; JAK/STAT signaling; Endocrinology/Hormones; Angiogenesis; Membrane transporter/Ion channel
Purity:
0.9957
SMILES:
CCC(=C(/c1ccc(O)cc1)c1ccc(OCCNC)cc1)c1ccccc1
Target:
Estrogen Receptor/ERR; EGFR; Potassium Channel; Estrogen/progestogen Receptor; HER

References

1. Chae YJ, et al. Eur J Pharmacol. 2015 Apr 5;752:1-7.2. Wu X, et al. Breast Y Res. 2011 Mar 10;13(2):R27.