TargetMol

SR 16832

Product Code:
 
TAR-T24827
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T24827-1mg1mg£177.00
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TAR-T24827-5mg5mg£313.00
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TAR-T24827-1mL1 mL * 10 mM (in DMSO)£322.00
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TAR-T24827-10mg10mg£430.00
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TAR-T24827-25mg25mg£663.00
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TAR-T24827-50mg50mg£863.00
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TAR-T24827-100mg100mg£1,179.00
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TAR-T24827-500mg500mg£2,311.00
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Further Information

Bioactivity:
SR 16832 is a dual-site PPARγ inhibitor. It also inhibits the binding of endogenous ligands and transcriptional activity of PPARγ, more effectively than the orthosteric covalent antagonist GW 9662 and T 0070907.
CAS:
2088135-12-8
Formula:
C17H12ClN3O4
Molecular Weight:
357.75
Pathway:
Metabolism; DNA Damage/DNA Repair
Purity:
0.98
SMILES:
COc1ccc2nccc(NC(=O)c3cc(ccc3Cl)[N+]([O-])=O)c2c1
Target:
PPAR

References

1. Brust et al (2017) Modification of the othosteric PPAR? covalent antagonist scaffold yields an improved dual-site allosteric inhibitor. ACS Chem.Biol. 12 969