TargetMol

RVX-297

Product Code:
 
TAR-T28628
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T28628-1mg1mg£138.00
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TAR-T28628-5mg5mg£229.00
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TAR-T28628-1mL1 mL * 10 mM (in DMSO)£252.00
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TAR-T28628-10mg10mg£334.00
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TAR-T28628-25mg25mg£519.00
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TAR-T28628-50mg50mg£703.00
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Quantity:
TAR-T28628-100mg100mg£970.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
RVX-297 is a BD2 selective inhibitor of BET bromodomains. RVX-297 preferentially binds to the BD2 domains of the BET bromodomain and Extra Terminal (BET) family of protein.
CAS:
1044871-04-6
Formula:
C24H29N3O4
Molecular Weight:
423.513
Pathway:
Chromatin/Epigenetic
Purity:
0.9811
SMILES:
COc1cc(OC)c2c(c1)nc([nH]c2=O)-c1cc(C)c(OCCN2CCCC2)c(C)c1
Target:
Epigenetic Reader Domain

References

1. Kharenko OA, et al. RVX-297- a novel BD2 selective inhibitor of BET bromodomains. Biochem Biophys Res Commun. 2016 Aug 12;477(1):62-7.