TargetMol

VPC171

Product Code:
 
TAR-T29112
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T29112-1mg1mg£160.00
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TAR-T29112-5mg5mg£250.00
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TAR-T29112-1mL1 mL * 10 mM (in DMSO)£253.00
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TAR-T29112-10mg10mg£327.00
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TAR-T29112-25mg25mg£544.00
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TAR-T29112-50mg50mg£744.00
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TAR-T29112-100mg100mg£1,002.00
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TAR-T29112-500mg500mg£1,942.00
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Further Information

Bioactivity:
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
CAS:
1018830-99-3
Formula:
C18H12F3NOS
Molecular Weight:
347.36
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.9952
SMILES:
Nc1scc(c1C(=O)c1ccccc1)-c1cccc(c1)C(F)(F)F
Target:
Adenosine Receptor

References

1. Aurelio L, et al. Allosteric modulators of the adenosine A1 receptor: synthesis and pharmacological evaluation of 4-substituted 2-amino-3-benzoylthiophenes. J Med Chem. 2009 Jul 23;52(14):4543-7. 2. Imlach WL, et al. A Positive Allosteric Modulator of the Adenosine A1 Receptor Selectively Inhibits Primary Afferent Synaptic Transmission in a Neuropathic Pain Model. Mol Pharmacol. 2015 Sep;88(3):460-8.