TargetMol

CAY10727

Product Code:
 
TAR-T36393
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T36393-5mg5mg£930.00
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TAR-T36393-50mg50mg£1,821.00
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Quantity:
TAR-T36393-100mg100mg£2,319.00
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This product comes from: United States.
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Further Information

Bioactivity:
CAY10727 is an inhibitor of protein arginine deiminase 3 (PAD3; kinact/KI= 15,600 M-1min-1).1It is selective for PAD3 over PAD1, -2, and -4 (kinact/KIs = 360, 1,110, and 1,460 M-1min-1, respectively).
CAS:
1671088-84-8
Formula:
C21H22Cl2N4O2
Molecular Weight:
433.3
Purity:
0.98
SMILES:
ClC1=CC=CC=C1C2=CC=CC(CN3C(NC(CCCNC(CCl)=N)C3=O)=O)=C2

References

Jamali, H., Khan, H.A., Stringer, J.R., et al.Identification of multiple structurally distinct, nonpeptidic small molecule inhibitors of protein arginine deiminase 3 using a substrate-based fragment methodJ. Am. Chem. Soc.137(10)3616-3621(2015)