TargetMol

DEPTOR-IN-1

Product Code:
 
TAR-T40242
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T40242-1mg1mg£182.00
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TAR-T40242-5mg5mg£349.00
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Quantity:
TAR-T40242-10mg10mg£516.00
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Quantity:
TAR-T40242-25mg25mg£791.00
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Quantity:
TAR-T40242-50mg50mg£1,058.00
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Quantity:
TAR-T40242-100mg100mg£1,396.00
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Quantity:
TAR-T40242-500mg500mg£2,713.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
DEPTOR-IN-1 is an inhibitor of DEPTOR with a Kd of 9.3 μM.
CAS:
2615911-12-9
Formula:
C24H16Cl2FNO4
Molecular Weight:
472.3
Purity:
0.9784
SMILES:
O=C1C(O)=C(C2=CC=C(Cl)C(Cl)=C2)OC3=C4CN(CC5=CC=CC(F)=C5)COC4=CC=C13

References

Hou Y, et al. Design, Synthesis, and Biological Evaluation of Icaritin Derivatives as Novel Putative DEPTOR Inhibitors for Multiple Myeloma Treatment. J Med Chem. 2021 Oct 28;64(20):14942-14954.