TargetMol

PZM21

Product Code:
 
TAR-T4386
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T4386-1mg1mg£106.00
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TAR-T4386-5mg5mg£148.00
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TAR-T4386-1mL1 mL * 10 mM (in DMSO)£164.00
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TAR-T4386-10mg10mg£205.00
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TAR-T4386-25mg25mg£309.00
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TAR-T4386-50mg50mg£483.00
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Quantity:
TAR-T4386-100mg100mg£670.00
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This product comes from: United States.
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Further Information

Bioactivity:
PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).
CAS:
1997387-43-5
Formula:
C19H27N3O2S
Molecular Weight:
361.5
Pathway:
Neuroscience; Endocrinology/Hormones; GPCR/G Protein
Purity:
0.9959
SMILES:
C[C@@H](Cc1ccsc1)NC(=O)NC[C@H](Cc1ccc(O)cc1)N(C)C
Target:
Opioid Receptor

References

Kostic M, et al. Biasing Opioid Receptors and Cholesterol as a Player in Developmental Biology. Manglik A, et al. Structure-based discovery of opioid analgesics with reduced side effects. Nature. 2016 Sep 8;537(7619):185-190.