TargetMol

DAMGO TFA (78123-71-4(Free base))

Product Code:
 
TAR-T4411
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T4411-1mg1mg£116.00
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TAR-T4411-2mg2mg£149.00
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TAR-T4411-5mg5mg£209.00
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TAR-T4411-10mg10mg£310.00
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TAR-T4411-25mg25mg£526.00
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TAR-T4411-50mg50mg£694.00
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Further Information

Bioactivity:
Potent, selective agonist of Mu-opioid receptor. Antinociceptive. Stimulates calcium-activated adenylyl cyclases related cAMP production. Expresses chemokines and chemokine receptors through TGF-beta1. Increases food intake of rats.
CAS:
T4411
Formula:
C28H36F3N5O8
Molecular Weight:
627.6
Pathway:
Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Purity:
0.9867
SMILES:
OC(=O)C(F)(F)F.C[C@@H](NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)NCC(=O)N(C)[C@@H](Cc1ccccc1)C(=O)NCCO
Target:
Opioid Receptor

References

Happel C,etal.DAMGO-induced expression of chemokines and chemokine receptors: the role of TGF-beta1.J Leukoc Biol. 2008 Apr;83(4):956-63. Onogi T,etal.DAMGO, a mu-opioid receptor selective agonist, distinguishes between mu- and delta-opioid receptors around their first extracellular loops.FEBS Lett. 1995 Jan 2;357(1):93-7. Rubovitch V,etal.The mu opioid agonist DAMGO stimulates cAMP production in SK-N-SH cells through a PLC-PKC-Ca++ pathway.Brain Res Mol Brain Res. 2003 Feb 20;110(2):261-6. Selve N,etal.Galanin receptor antagonists attenuate spinal antinociceptive effects of DAMGO, tramadol and non-opioid drugs in rats.Brain Res. 1996 Oct 7;735(2):177-87. Szab? G,etal.Long-lasting antinociceptive effect of DAMGO chloromethyl ketone in rats.Peptides. 1999 Nov;20(11):1321-6.