TargetMol

SGC-GAK-1

Product Code:
 
TAR-T5169
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T5169-1mg1mg£95.00
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TAR-T5169-5mg5mg£128.00
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TAR-T5169-1mL1 mL * 10 mM (in DMSO)£134.00
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TAR-T5169-10mg10mg£168.00
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TAR-T5169-25mg25mg£269.00
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TAR-T5169-50mg50mg£389.00
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Quantity:
TAR-T5169-100mg100mg£544.00
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This product comes from: United States.
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Further Information

Bioactivity:
SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).
CAS:
2226517-76-4
Formula:
C18H17BrN2O3
Molecular Weight:
389.249
Pathway:
Metabolism; Cell Cycle/Checkpoint
Purity:
0.9974
SMILES:
COc1cc(Nc2ccnc3ccc(Br)cc23)cc(OC)c1OC
Target:
Serine/threonin kinase

References

Asquith CRM, et al. SGC-GAK-1: A Chemical Probe for Cyclin G Associated Kinase (GAK). J Med Chem. 2019 Feb 26.