TargetMol

Branebrutinib

Product Code:
 
TAR-T5407
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T5407-1mg1mg£114.00
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TAR-T5407-1mL1 mL * 10 mM (in DMSO)£193.00
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TAR-T5407-5mg5mg£193.00
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TAR-T5407-10mg10mg£258.00
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TAR-T5407-25mg25mg£386.00
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TAR-T5407-50mg50mg£539.00
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TAR-T5407-100mg100mg£741.00
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TAR-T5407-200mg200mg£994.00
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Quantity:
TAR-T5407-500mg500mg£1,428.00
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Further Information

Bioactivity:
BMS986195 is a potent, covalent inhibitor of Bruton's tyrosine kinase (BTK), >5,000-fold selective over all kinases outside of the Tec family (IC50 <1 nM for BTK).
CAS:
1912445-55-6
Formula:
C20H23FN4O2
Molecular Weight:
370.428
Pathway:
Tyrosine Kinase/Adaptors; Angiogenesis
Purity:
0.9939
SMILES:
CC#CC(=O)N[C@H]1CCCN(C1)c1c(F)cc(C(N)=O)c2[nH]c(C)c(C)c12
Target:
BTK

References

JR Burke, et al. BMS-986195 Is a Highly Selective and Rapidly Acting Covalent Inhibitor of Bruton?s Tyrosine Kinase with Robust Efficacy at Low Doses in Preclinical Models of RA and Lupus Nephritis. 2017 ACR/ARHP Annual Meeting, September 18, 2017.