TargetMol

TAPI1

Product Code:
 
TAR-T6009
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
 

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CodeSizePrice
TAR-T6009-1mg1mg£229.00
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TAR-T6009-2mg2mg£335.00
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TAR-T6009-1mL1 mL * 10 mM (in DMSO)£573.00
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TAR-T6009-5mg5mg£573.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
TAPI-1, an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.
CAS:
163847-77-6
Formula:
C26H37N5O5
Molecular Weight:
499.612
Pathway:
Proteases/Proteasome
Purity:
0.98
SMILES:
CC(C)CC(CC(=O)NO)C(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C)C(=O)NCCN
Target:
MMP

References

Slack BE, et al. Biochem J. 2001, 357(Pt 3), 787-794. M?llberg J, et al. J Immunol. 1995, 155(11), 5198-5205 Sisto M, et al. 2014. DOI 10.12007/s10238-2014-0279-4. Oikawa H, et al. Life Sci. 2014, 97(2), 137-144.