TargetMol

A-836339

Product Code:
 
TAR-T7375
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7375-1mg1mg£102.00
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TAR-T7375-1mL1 mL * 10 mM (in DMSO)£185.00
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TAR-T7375-5mg5mg£195.00
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TAR-T7375-10mg10mg£294.00
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TAR-T7375-25mg25mg£446.00
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TAR-T7375-50mg50mg£623.00
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TAR-T7375-100mg100mg£856.00
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Further Information

Bioactivity:
A-836339 acts as a potent cannabinoid receptor full agonist which has a higher affinity for the peripheral CB2 receptor (Ki = 0.64 nM) over the central CB1 receptor (Ki = 270 nM). It displays analgesic, anti-inflammatory, and anti-hyperalgesic effects in mice.
CAS:
959746-77-1
Formula:
C16H26N2O2S
Molecular Weight:
310.46
Pathway:
GPCR/G Protein
Purity:
0.98
SMILES:
COCCn1c(C)c(C)sc1=NC(=O)C1C(C)(C)C1(C)C
Target:
Cannabinoid Receptor

References

Characterization of a Cannabinoid CB2 Receptor-Selective Agonist, A-836339 [2,2,3,3-Tetramethyl-cyclopropanecarboxylic Acid [3-(2-Methoxy-ethyl)-4,5-dimethyl-3H-thiazol-(2Z)-ylidene]-amide], Using in Vitro Pharmacological Assays, in Vivo Pain Models, and Pharmacological Magnetic Resonance Imaging[J]. Journal of Pharmacology and Experimental Therapeutics, 2009, 328(1):141-151. Mcgaraughty S , Chu K M , Yao B , et al. A CB 2, receptor agonist, A-836339, modulates wide dynamic range neuronal activity in neuropathic rats: Contributions of spinal and peripheral CB 2, receptors[J]. Neuroscience, 2009, 158(4):1652-1661.