TargetMol

Deltorphin 2

Product Code:
 
TAR-T7639
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7639-1mg1mg£116.00
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TAR-T7639-5mg5mg£213.00
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TAR-T7639-10mg10mg£333.00
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TAR-T7639-25mg25mg£516.00
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TAR-T7639-50mg50mg£711.00
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TAR-T7639-100mg100mg£946.00
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This product comes from: United States.
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Further Information

Bioactivity:
Deltorphin 2(TFA) is an agonist of δ opioid receptor(IC50:0.41 nM)
CAS:
122752-16-3
Formula:
C38H54N8O10
Molecular Weight:
782.896
Pathway:
GPCR/G Protein; Endocrinology/Hormones; Neuroscience
Purity:
1
SMILES:
CC(C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(C)C)C(=O)NCC(N)=O
Target:
Opioid Receptor

References

Thomas S A , Abbruscato T J , Hau V S , et al. Structure-Activity Relationships of a Series of [D-Ala2]Deltorphin I and II Analogues ;[J]. Journal of Pharmacology and Experimental Therapeutics, 1997, 281(2):817-825. Willemse T, et al. Chemical space screening around Phe3 in opioid peptides: Modulating ? versus ? agonism by Suzuki-Miyaura cross-couplings. Bioorg Med Chem Lett. 2018 Jul 15;28(13):2320-2323. doi: 10.1016/j.bmcl.2018.05.015. Epub 2018 May 12. Erratum in: Bioorg Med Chem Lett. 2018 Nov 1;28(20):3418.