TargetMol

LML134

Product Code:
 
TAR-T8514
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T8514-1mg1mg£179.00
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TAR-T8514-2mg2mg£226.00
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TAR-T8514-1mL1 mL * 10 mM (in DMSO)£283.00
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TAR-T8514-5mg5mg£301.00
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TAR-T8514-10mg10mg£436.00
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TAR-T8514-25mg25mg£675.00
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TAR-T8514-50mg50mg£922.00
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TAR-T8514-100mg100mg£1,219.00
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This product comes from: United States.
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Further Information

Bioactivity:
LML-134 is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).
CAS:
1542135-76-1
Formula:
C19H29N5O3
Molecular Weight:
375.473
Pathway:
Immunology/Inflammation; Neuroscience; GPCR/G Protein
Purity:
0.9986
SMILES:
Cn1nc(ccc1=O)N1CCC(CC1)OC(=O)N1CCN(CC1)C1CCC1
Target:
Histamine Receptor

References

Troxler T, et al. The Discovery of LML134, a Histamine H3 Receptor Inverse Agonist for the Clinical Treatment of Excessive Sleep Disorders. ChemMedChem. 2019 Jul 3;14(13):1238-1247.