TargetMol

Desketoraloxifene

Product Code:
 
TAR-T9001
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T9001-5mg5mg£313.00
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TAR-T9001-10mg10mg£435.00
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TAR-T9001-25mg25mg£728.00
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This product comes from: United States.
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Further Information

Bioactivity:
Desketoraloxifene is a selective estrogen receptor modulator, inhibiting mammalian PLD (PLD1 and PLD2).
CAS:
216570-81-9
Formula:
C27H27NO3S
Molecular Weight:
445.57
Pathway:
Metabolism
Purity:
0.98
SMILES:
C1CCN(CC1)CCOC2=CC=C(C=C2)C3=C(SC4=C3C=CC(=C4)O)C5=CC=C(C=C5)O
Target:
Phospholipase

References

Scott S A , Spencer C T , MC O?Reilly, et al. Discovery of Desketoraloxifene Analogues as Inhibitorsof Mammalian, Pseudomonas aeruginosa, and NAPE PhospholipaseD Enzymes[J]. Acs Chemical Biology, 2015, 10(2):421. Cho C H , Jung D I , Neuenswander B , et al. Parallel synthesis of a desketoraloxifene analogue library via iodocyclization/palladium-catalyzed coupling.[J]. Acs Combinatorial Science, 2011, 13(5):501-510.