TargetMol

CHR-6494 TFA

Product Code:
 
TAR-T9521
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T9521-1mg1mg£148.00
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TAR-T9521-2mg2mg£189.00
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TAR-T9521-5mg5mg£245.00
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TAR-T9521-1mL1 mL * 10 mM (in DMSO)£275.00
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TAR-T9521-10mg10mg£353.00
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TAR-T9521-25mg25mg£544.00
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Quantity:
TAR-T9521-50mg50mg£744.00
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TAR-T9521-100mg100mg£1,002.00
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Quantity:
TAR-T9521-500mg500mg£1,942.00
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This product comes from: United States.
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Further Information

Bioactivity:
CHR-6494 TFA is a potent haspin inhibitor, with an?IC50?of 2 nM. It inhibits histone H3T3 phosphorylation. CHR-6494 TFA induces the?apoptosis?of cancer cells, including melanoma and breast cancer. CHR-6494 TFA can be used in the research of cancer
CAS:
1458630-17-5
Formula:
C18H17F3N6O2
Molecular Weight:
406.362
Purity:
0.991
SMILES:
OC(=O)C(F)(F)F.CCCNc1ccc2ncc(-c3ccc4[nH]ncc4c3)n2n1

References

Huertas D, et al. Antitumor activity of a small-molecule inhibitor of the histone kinase Haspin. Oncogene. 2012 Mar 15;31(11):1408-18.