TargetMol

TRPM8 antagonist 3

Product Code:
 
TAR-T9709
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T9709-1mg1mg£145.00
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TAR-T9709-5mg5mg£254.00
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Quantity:
TAR-T9709-1mL1 mL * 10 mM (in DMSO)£274.00
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TAR-T9709-10mg10mg£356.00
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TAR-T9709-25mg25mg£544.00
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TAR-T9709-50mg50mg£760.00
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Quantity:
TAR-T9709-100mg100mg£1,018.00
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This product comes from: United States.
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Further Information

Bioactivity:
TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).
CAS:
2102179-29-1
Formula:
C13H12N2O4S
Molecular Weight:
292.315
Pathway:
Membrane transporter/Ion channel
Purity:
0.9925
SMILES:
O=C(C1=C(O)N=C(C2=CC=CC=C2O)S1)N3OCCC3
Target:
TRP/TRPV Channel

References

Bianchini G, et al. Discovery of Novel TRPM8 Blockers Suitable for the Treatment of Somatic and Ocular Painful Conditions: A Journey through pKa and LogD Modulation. J Med Chem. 2021 Nov 25;64(22):16820-16837.