TargetMol

SETDB1-TTD-IN-1

Product Code:
 
TAR-T9742
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T9742-1mg1mg£287.00
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TAR-T9742-5mg5mg£605.00
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TAR-T9742-1mL1 mL * 10 mM (in DMSO)£699.00
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TAR-T9742-10mg10mg£832.00
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TAR-T9742-25mg25mg£1,211.00
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TAR-T9742-50mg50mg£1,589.00
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Quantity:
TAR-T9742-100mg100mg£2,135.00
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This product comes from: United States.
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Further Information

Bioactivity:
SETDB1-TTD-IN-1 is a potent, selective and endogenous binder competitive inhibitor of SETDB1-TTD with a Kd of 88 nM.
CAS:
2755823-12-0
Formula:
C28H31N5O2
Molecular Weight:
469.58
Pathway:
Chromatin/Epigenetic
Purity:
0.98
SMILES:
CN1C[C@H](C[C@H](C1)NC2=NC3=C(NC=C3)C(N2CC=C)=O)C4=CC=C(C=C4)OCC5=CC=CC=C5
Target:
Histone Methyltransferase

References

Guo Y, et, al. Structure-Guided Discovery of a Potent and Selective Cell-Active Inhibitor of SETDB1 Tudor Domain. Angew Chem Int Ed Engl. 2021 Apr 12;60(16):8760-8765.