TargetMol

Opiranserin hydrochloride

Product Code:
 
TAR-T9833
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T9833-1mg1mg£164.00
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TAR-T9833-5mg5mg£303.00
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TAR-T9833-1mL1 mL * 10 mM (in DMSO)£326.00
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TAR-T9833-10mg10mg£442.00
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TAR-T9833-25mg25mg£686.00
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TAR-T9833-50mg50mg£930.00
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TAR-T9833-100mg100mg£1,235.00
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TAR-T9833-500mg500mg£2,384.00
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This product comes from: United States.
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Further Information

Bioactivity:
Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM, respectively. It shows antagonistic activity on rP2X3 (IC50=0.87 μM). It is development as an injectable agent for the treatment of postoperative pain.
CAS:
1440796-75-7
Formula:
C21H35ClN2O5
Molecular Weight:
430.97
Pathway:
GPCR/G Protein; Neuroscience; Membrane transporter/Ion channel
Purity:
0.98
SMILES:
O=C(NCC1(N(C)C)CCOCC1)C2=CC(OC)=C(OCCCC)C(OC)=C2.[H]Cl
Target:
P2X Receptor; GlyT; 5-HT Receptor