TargetMol

PARP1-IN-8?

Product Code:
 
TAR-T9891
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T9891-1mg1mg£148.00
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TAR-T9891-5mg5mg£269.00
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TAR-T9891-1mL1 mL * 10 mM (in DMSO)£301.00
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TAR-T9891-10mg10mg£389.00
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TAR-T9891-25mg25mg£603.00
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TAR-T9891-50mg50mg£830.00
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Quantity:
TAR-T9891-100mg100mg£1,099.00
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Quantity:
TAR-T9891-500mg500mg£2,135.00
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This product comes from: United States.
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Further Information

Bioactivity:
PARP1-IN-8 is an effective inhibito of PARP1 (IC50 = 97 nM).
CAS:
836640-15-4
Formula:
C23H18ClN3O2
Molecular Weight:
403.87
Pathway:
DNA Damage/DNA Repair; Chromatin/Epigenetic
Purity:
0.9826
SMILES:
Clc1cccc(NC(=O)CCn2nc(-c3ccccc3)c3ccccc3c2=O)c1
Target:
PARP

References

Almahli H, Hadchity E, Jaballah MY, Daher R, Ghabbour HA, Kabil MM, Al-Shakliah NS, Eldehna WM. Development of novel synthesized phthalazinone-based PARP-1 inhibitors with apoptosis inducing mechanism in lung cancer. Bioorg Chem. 2018 Apr;77:443-456.