TargetMol

GLL 398

Product Code:
 
TAR-T9997
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T9997-1mg1mg£227.00
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TAR-T9997-5mg5mg£422.00
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TAR-T9997-1mL1 mL * 10 mM (in DMSO)£430.00
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TAR-T9997-10mg10mg£597.00
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TAR-T9997-25mg25mg£1,017.00
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Quantity:
TAR-T9997-50mg50mg£1,491.00
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Quantity:
TAR-T9997-100mg100mg£2,201.00
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Quantity:
TAR-T9997-200mg200mg£3,266.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GLL 398 is an orally active and selective degrader of estrogen receptor with an IC50 of 1.14 nM. GLL 398 blocks tumor growth in xenograft breast cancer models.
CAS:
2077980-80-2
Formula:
0
Molecular Weight:
0
Pathway:
Endocrinology/Hormones
Purity:
0.98
SMILES:
0
Target:
Estrogen Receptor/ERR

References

Guo S, et al. GLL398, an oral selective estrogen receptor degrader (SERD), blocks tumor growth in xenograft breast cancer models. Breast Cancer Res Treat. 2020;180(2):359-368.