TargetMol

PKG Substrate acetate?81187-14-6 free base)

Product Code:
 
TAR-TP1787L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-TP1787L-1mg1mg£152.00
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Quantity:
TAR-TP1787L-5mg5mg£365.00
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TAR-TP1787L-10mg10mg£511.00
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TAR-TP1787L-25mg25mg£782.00
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Quantity:
TAR-TP1787L-50mg50mg£1,026.00
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Quantity:
TAR-TP1787L-100mg100mg£1,380.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PKG Substrate acetate is a selective substrate for cGMP-dependent protein kinase (PKG).PKG Substrate is a selective substrate for protein kinase G (PKG) with a strong preference for PKG Iα (Km = 59 μM) over PKG II (Km = 305 μM).
CAS:
TP1787L
Formula:
C37H71N17O13
Molecular Weight:
962.08
Pathway:
Tyrosine Kinase/Adaptors
Purity:
0.993
SMILES:
CC(O)=O.O=C(O)CC[C@@H](C(O)=O)NC([C@H](C)NC([C@H](CCCNC(N)=N)NC([C@H](CO)NC([C@H](CCCNC(N)=N)NC([C@H](CCCCN)NC([C@H](CCCNC(N)=N)N)=O)=O)=O)=O)=O)=O
Target:
PKA

References

Wong A, et al. Cyclic GMP-dependent stimulation of serotonin transport does not involve direct transporter phosphorylation by cGMP-dependent protein kinase. J Biol Chem. 2012 Oct 19;287(43):36051-8.