TargetMol

Orphanin FQ(1-11) acetate(178249-41-7 free base)

Product Code:
 
TAR-TP1882L1
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-TP1882L1-1mg1mg£201.00
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TAR-TP1882L1-5mg5mg£364.00
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TAR-TP1882L1-10mg10mg£510.00
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TAR-TP1882L1-25mg25mg£780.00
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TAR-TP1882L1-50mg50mg£1,026.00
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TAR-TP1882L1-100mg100mg£1,380.00
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Further Information

Bioactivity:
Peptide fragment containing amino acids 1-11 of Nociceptin. Potent agonist of the ORL1/KOR-3 receptor (Ki = 55 nM); displays no affinity for opioid receptors, including μ, δ, κ1 and κ3 receptors (Ki >1000 nM). Displays analgesic properties in CD-1 mice.
CAS:
TP1882L1
Formula:
C51H79N15O16
Molecular Weight:
1158.26
Pathway:
GPCR/G Protein; Endocrinology/Hormones; Neuroscience
Purity:
0.9554
SMILES:
0
Target:
Opioid Receptor

References

Rossi et al (1997) Pharmacological characterization of orphanin FQ/nociceptin and its fragments. J.Pharmacol.Exp.Ther. 282 858 PMID: Rossi et al (1998) Orphanin FQ/nociceptin analgesia in the rat. Brain Res. 792 327 PMID: Reinscheid et al (1996) Structure-activity relationship studies on the novel neuropeptide orphanin FQ. J.Biol.Chem. 271 14163 PMID: