TargetMol

MLCK inhibitor peptide 18

Product Code:
 
TAR-TP1890
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TP1890-1mg1mg£113.00
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TAR-TP1890-5mg5mg£210.00
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TAR-TP1890-10mg10mg£324.00
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Quantity:
TAR-TP1890-25mg25mg£635.00
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This product comes from: United States.
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Further Information

Bioactivity:
Selective competitive inhibitor of myosin light chain kinase (IC50 = 50 nM). Displays 4000-fold selectivity over CaM kinase II and does not inhibit PKA. Cell permeable.
CAS:
224579-74-2
Formula:
C60H105N23O11
Molecular Weight:
1324.64
Purity:
0.98
SMILES:
0

References

Lukas et al (1999) Identification of novel classes of protein kinase inhibitors using combinatorial peptide chemistry based on functional genomics knowledge. J.Med.Chem. 42 910 PMID: Zolotarevsky et al (2002) A membrane-permeant peptide that inhibits MLC kinase restores barrier function in in vitro models of intestinal disease. Gastroenterology 123 163 PMID: