TargetMol

G-Protein antagonist peptide acetate

Product Code:
 
TAR-TP1902L1
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TP1902L1-1mg1mg£182.00
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TAR-TP1902L1-2mg2mg£258.00
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TAR-TP1902L1-5mg5mg£364.00
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TAR-TP1902L1-10mg10mg£537.00
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TAR-TP1902L1-25mg25mg£809.00
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TAR-TP1902L1-50mg50mg£1,075.00
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Quantity:
TAR-TP1902L1-100mg100mg£1,428.00
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Further Information

Bioactivity:
G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide acetate inhibits the activation of Gi or Go by M2 muscarinic cholinergic receptor (M2 mAChR) or of Gs by beta-adrenergic receptor in the reconstituted phospholipid vesicles, assayed by receptor-promoted GTP hydrolysis
CAS:
TP1902L1
Formula:
C59H68N12O11S
Molecular Weight:
1153.33
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.9806
SMILES:
CSCC[C@@H](C(N)=O)NC([C@@H](CC1=CNC2=CC=CC=C12)NC([C@H](NC([C@H](CC3=CC=CC=C3)NC([C@H](NC([C@H](CCC(N)=O)NC([C@H]4NC(CC4)=O)=O)=O)CC5=CNC6=CC=CC=C56)=O)=O)CC7=CNC8=CC=CC=C78)=O)=O.CC(O)=O
Target:
Adrenergic Receptor

References

Mukai H, et al. G protein antagonists. A novel hydrophobic peptide competes with receptor for G protein binding. J Biol Chem. 1992;267(23):16237-16243.