TargetMol

ELA-14(human) acetate

Product Code:
 
TAR-TP1923L1
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
 

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CodeSizePrice
TAR-TP1923L1-1mg1mg£147.00
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TAR-TP1923L1-5mg5mg£356.00
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TAR-TP1923L1-10mg10mg£499.00
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TAR-TP1923L1-25mg25mg£764.00
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TAR-TP1923L1-50mg50mg£1,026.00
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TAR-TP1923L1-100mg100mg£1,340.00
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This product comes from: United States.
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Further Information

Bioactivity:
ELA-14(human) acetate is a fragment of ELA that binds to APJ, activates the Gαi1 and β-arrestin-2 signaling pathways, and induces receptor internalization similarly to its parent endogenous peptide.
CAS:
TP1923L1
Formula:
C77H123N25O19S2
Molecular Weight:
1767.09
Pathway:
GPCR/G Protein
Purity:
0.98
SMILES:
CC(C)C[C@@H](C(N[C@@H](Cc1c[nH]cn1)C(N[C@@H](CO)C(N[C@@H](CCCNC(N)=N)C(N[C@@H](C(C)C)C(N(CCC1)[C@@H]1C(N[C@@H](Cc1ccccc1)C(N(CCC1)[C@@H]1C(O)=O)=O)=O)=O)=O)=O)=O)=O)NC([C@H](CCC1)N1C([C@H](CCSC)NC([C@H](CS)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC([C@H](
Target:
Apelin receptor

References

Alexandre Murza, et al. Discovery and Structure-Activity Relationship of a Bioactive Fragment of ELABELA That Modulates Vascular and Cardiac Functions. J Med Chem. 2016 Apr 14;59(7):2962-72.