TargetMol

WRW4 TFA(878557-55-2 free base)

Product Code:
 
TAR-TP1926
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TP1926-1mg1mg£139.00
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Quantity:
TAR-TP1926-5mg5mg£224.00
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Quantity:
TAR-TP1926-10mg10mg£302.00
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Quantity:
TAR-TP1926-25mg25mg£484.00
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Quantity:
TAR-TP1926-50mg50mg£670.00
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Quantity:
TAR-TP1926-100mg100mg£914.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
WRW4 is a specific formyl peptide receptor-like 1 (FPRL1) antagonist, inhibits WKYMVm binding to FPRL1 with an IC50 of 0.23 μM. WRW4 specifically inhibits the increase in intracellular calcium by the FPRL1 agonists MMK-1, amyloid beta42 (Abeta42) peptide, and F peptide.
CAS:
TP1926
Formula:
C63H66F3N15O8
Molecular Weight:
1218.29
Purity:
0.999
SMILES:
C1=CC=C2C(=C1)C(=CN2)C[C@@H](C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC3=CNC4=CC=CC=C43)C(=O)N[C@@H](CC5=CNC6=CC=CC=C65)C(=O)N[C@@H](CC7=CNC8=CC=CC=C87)C(=O)N[C@@H](CC9=CNC1=CC=CC=C19)C(=O)N)N.OC(C(F)(F)F)=O

References

Bae et al (2004) Identification of peptides that antagonize formyl peptide receptor-like 1-mediating signaling. J.Immunol. 173 607 PMID: