TargetMol

PG 106 acetate

Product Code:
 
TAR-TP1952L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
 

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CodeSizePrice
TAR-TP1952L-1mg1mg£212.00
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TAR-TP1952L-5mg5mg£550.00
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TAR-TP1952L-10mg10mg£755.00
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TAR-TP1952L-25mg25mg£1,107.00
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TAR-TP1952L-50mg50mg£1,460.00
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Quantity:
TAR-TP1952L-100mg100mg£1,958.00
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This product comes from: United States.
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Further Information

Bioactivity:
PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with the hMC5 receptor and hMC4 receptors with an EC50 of 9900 nM.
CAS:
0
Formula:
C53H73N13O11
Molecular Weight:
1068.23
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.9824
SMILES:
CCCCC(NC(C)=O)C(N[C@H]1CC(NCCCC[C@@H](C(N)=O)NC([C@H](CC2=CNC3=CC=CC=C32)NC([C@H](CCC/N=C(N)N)NC([C@@H](CC4=CC5=CC=CC=C5C=C4)NC(CCNC1=O)=O)=O)=O)=O)=O)=O.CC(O)=O
Target:
Melanocortin Receptor

References

Paolo Grieco, et al. Further structure-activity studies of lactam derivatives of MT-II and SHU-9119: their activity and selectivity at human melanocortin receptors 3, 4, and 5. Peptides