TargetMol

PKI (5-24) Acetate(99534-03-9 free base)

Product Code:
 
TAR-TP1957L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TP1957L-1mg1mg£177.00
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Quantity:
TAR-TP1957L-5mg5mg£287.00
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Quantity:
TAR-TP1957L-10mg10mg£438.00
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TAR-TP1957L-25mg25mg£675.00
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Quantity:
TAR-TP1957L-50mg50mg£922.00
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Quantity:
TAR-TP1957L-100mg100mg£1,219.00
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Quantity:
TAR-TP1957L-500mg500mg£2,368.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PKI (5-24) Acetate is a high affinity PKA inhibitor (Ki = 2.3 nM).
CAS:
TP1957L
Formula:
C96H152N32O33
Molecular Weight:
2282.43
Pathway:
Tyrosine Kinase/Adaptors
Purity:
0.9947
SMILES:
0
Target:
PKA

References

Cheng et al (1986) A potent synthetic peptide inhibitor of the cAMP-dependent protein kinase. J.Biol.Chem. 261 989 PMID: Narayana et al (1997) Crystal structure of a polyhistidine-tagged recombinant catalytic subunit of cAMP-dependent protein kinase complexed with the peptide inhibitor PKI(5-24) and adenosine. Biochemistry 36 4438 PMID: