TargetMol

BigLEN (mouse) acetate

Product Code:
 
TAR-TP2073L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
 

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CodeSizePrice
TAR-TP2073L-1mg1mg£189.00
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TAR-TP2073L-5mg5mg£340.00
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TAR-TP2073L-10mg10mg£470.00
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TAR-TP2073L-25mg25mg£707.00
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TAR-TP2073L-50mg50mg£978.00
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TAR-TP2073L-100mg100mg£1,291.00
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Further Information

Bioactivity:
BigLEN (mouse) acetate is a potent and selective agonist of orphan G protein-coupled receptor 171 (GPR171), with a Kd of ?0.5 nM.
CAS:
TP2073L
Formula:
C80H134N24O24
Molecular Weight:
1816.07
Pathway:
GPCR/G Protein; Endocrinology/Hormones
Purity:
0.9834
SMILES:
O=C(O)[C@H]1N(C([C@H]2N(C([C@H](CC(C)C)NC([C@H](CC(C)C)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC([C@H](C)NC([C@H]3N(C([C@H](C)NC([C@H](CCC(N)=O)NC([C@H]4N(C([C@H](CO)NC([C@H]5N(C([C@H](CC(N)=O)NC([C@H](CCC(O)=O)NC([C@H](CC(C)C)N)=O)=O)=O)CCC5)=O)=O)CCC4)=O)=O)=O)CCC3)=O)=O)=O)=O)=O)=O)CCC2)=O)CCC1.CC(O)=O
Target:
GPR

References

Gomes I, et, al. GPR171 is a hypothalamic G protein-coupled receptor for BigLEN, a neuropeptide involved in feeding. Proc Natl Acad Sci U S A. 2013 Oct 1;110(40):16211-6. Mack SM, et, al. Neuropeptide PEN and Its Receptor GPR83: Distribution, Signaling, and Regulation. ACS Chem Neurosci. 2019 Apr 17;10(4):1884-1891.