TargetMol

Fulacimstat

Product Code:
 
TAR-TQ0035
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TQ0035-1mg1mg£179.00
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TAR-TQ0035-5mg5mg£303.00
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TAR-TQ0035-1mL1 mL * 10 mM (in DMSO)£309.00
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TAR-TQ0035-10mg10mg£402.00
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TAR-TQ0035-25mg25mg£626.00
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TAR-TQ0035-50mg50mg£862.00
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Quantity:
TAR-TQ0035-100mg100mg£1,139.00
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This product comes from: United States.
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Further Information

Bioactivity:
Fulacimstat (BAY1142524) is a chymase inhibitor, with IC50s of 3, 4 nM for hamster and human chymase enzyme, respectively.
CAS:
1488354-15-9
Formula:
C23H16F3N3O6
Molecular Weight:
487.391
Purity:
0.9977
SMILES:
Cn1c2ccc(cc2oc1=O)-n1cc(C(O)=O)c(=O)n([C@@H]2CCc3c2cccc3C(F)(F)F)c1=O

References

Hanna Tinel, et al. Abstract 13624: A Novel Chymase Inhibitor BAY 1142524 Reduces Fibrosis and Improves Cardiac Function After Myocardial Infarction in Hamster. Circulation. 2018;136:A13624.